Molecule Details
InChIKeyWRJITTKUXGEQBF-KJKBHKFMSA-N
Compound NameArchazolid F
Canonical SMILESCNC(=O)O[C@@H](CC(C)C)c1nc([C@H]2OC(=O)C/C=C/C(C)=C/[C@@H](O)[C@@H](C)/C=C(C)\C=C(C)/C=C/[C@@H](O)[C@H](C)[C@H](OC)/C(C)=C/C=C/[C@@H]2C)cs1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.17
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P56373 P2RX3 Homo sapiens Human PF00864 6.4 IC50 ChEMBL;BindingDB
P08246 ELANE Homo sapiens Human PF00089 6.1 IC50 ChEMBL;BindingDB
P0DMS8 ADORA3 Homo sapiens Human PF00001 6.1 Ki ChEMBL;BindingDB