Molecule Details
InChIKeyWPOYFQFVGWXOSQ-UHFFFAOYSA-N
Compound NameN-[3-[(6-chloro-1,2,3,4-tetrahydroacridin-9-yl)amino]propyl]-2-[2-(cyclopropanecarbonylamino)-4-pyridinyl]-4-methoxy-1,3-thiazole-5-carboxamide
Canonical SMILESCOc1nc(-c2ccnc(NC(=O)C3CC3)c2)sc1C(=O)NCCCNc1c2c(nc3cc(Cl)ccc13)CCCC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.72
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P22303 ACHE Homo sapiens Human PF08674 PF00135 8.4 IC50 ChEMBL;BindingDB
P49841 GSK3B Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB