Molecule Details
InChIKeyWPLZOHYVBARFAX-GFCCVEGCSA-N
Compound Name2-oxo-3-[(1R)-1-(1,2,3,4-tetrahydroisoquinolin-8-yl)ethyl]-N-(1,2,4-thiadiazol-5-yl)-1,3-benzoxazole-6-sulfonamide
Canonical SMILESC[C@H](c1cccc2c1CNCC2)n1c(=O)oc2cc(S(=O)(=O)Nc3ncns3)ccc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.57
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15858 SCN9A Homo sapiens Human PF00520 PF24609 PF06512 PF11933 7.6 IC50 ChEMBL;BindingDB
Q99250 SCN2A Homo sapiens Human PF00520 PF24609 PF06512 PF11933 7.5 IC50 ChEMBL;BindingDB