Molecule Details
InChIKeyWPHLFVIDUSHWHQ-UHFFFAOYSA-N
Compound Name4-(6-(2-chlorophenylamino)-1H-indazol-3-yl)-N-(2-(dimethylamino)ethyl)benzamide
Canonical SMILESCN(C)CCNC(=O)c1ccc(-c2n[nH]c3cc(Nc4ccccc4Cl)ccc23)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.04
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P53779 MAPK10 Homo sapiens Human PF00069 8.7 IC50 ChEMBL;BindingDB
Q16539 MAPK14 Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB
P45983 MAPK8 Homo sapiens Human PF00069 7.3 IC50 ChEMBL;BindingDB