Molecule Details
InChIKeyWOTGMDIMMYQXRU-UHFFFAOYSA-N
Canonical SMILESCC(=O)Nc1ccc(S(=O)(=O)N(Cc2c[nH]nn2)c2ccc(N(Cc3c[nH]nn3)S(=O)(=O)c3ccc(NC(C)=O)cc3)c3ccccc23)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.21
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16236 NFE2L2 Homo sapiens Human PF03131 6.2 IC50 ChEMBL;BindingDB
Q14145 KEAP1 Homo sapiens Human PF07707 PF00651 PF01344 PF24681 6.2 IC50 ChEMBL