Molecule Details
InChIKeyWOSWUKXUZVAPGM-UHFFFAOYSA-N
Compound NameN-(2-methoxyquinolin-6-yl)-3-propan-2-yl-2,5,11,13-tetrazatricyclo[7.4.0.02,6]trideca-1(13),3,5,7,9,11-hexaen-12-amine
Canonical SMILESCOc1ccc2cc(Nc3ncc4ccc5ncc(C(C)C)n5c4n3)ccc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.12
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB
P24385 CCND1 Homo sapiens Human PF02984 PF00134 7.1 IC50 ChEMBL;BindingDB
Q00534 CDK6 Homo sapiens Human PF00069 7.1 IC50 ChEMBL