Molecule Details
InChIKeyWOEBXQWHXAFLRS-UHFFFAOYSA-N
Compound Name3-[2-(2-amino-1,1-difluoroethyl)-1H-benzimidazol-4-yl]-6-(2-aminoethylsulfonyl)-2-(2H-tetrazol-5-yl)benzenesulfonamide
Canonical SMILESNCCS(=O)(=O)c1ccc(-c2cccc3[nH]c(C(F)(F)CN)nc23)c(-c2nn[nH]n2)c1S(N)(=O)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL10.33
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9XAY4 blaVIM Pseudomonas aeruginosa Pathogen PF00753 10.5 IC50 BindingDB
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 10.4 IC50 ChEMBL;BindingDB
P52699 Serratia marcescens Pathogen PF00753 10.1 IC50 BindingDB