Molecule Details
InChIKeyWNTHBRVKPVTIQB-UHFFFAOYSA-N
Compound NameMethyl 6-bromo-2-[(4-methanesulfonylphenyl)methyl]-1-oxo-4-phenyl-1,2-dihydroisoquinoline-3-carboxylate
Canonical SMILESCOC(=O)c1c(-c2ccccc2)c2cc(Br)ccc2c(=O)n1Cc1ccc(S(C)(=O)=O)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.5
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB