Molecule Details
InChIKeyWNMOTZHMKYYWSU-UHFFFAOYSA-N
Compound Name3-chloro-N-methyl-4-(5-(1-methyl-1H-pyrazol-4-yl)-4-(tetrahydro-2H-pyran-4-yloxy)-7H-pyrrolo[2,3-d]pyrimidin-2-ylamino)benzamide
Canonical SMILESCNC(=O)c1ccc(Nc2nc(OC3CCOCC3)c3c(-c4cnn(C)c4)c[nH]c3n2)c(Cl)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.07
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P33981 TTK Homo sapiens Human PF00069 8.7 IC50 ChEMBL;BindingDB
P49760 CLK2 Homo sapiens Human PF00069 8.5 IC50 ChEMBL;BindingDB
P49759 CLK1 Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB