Molecule Details
InChIKeyWLXUDQMWNQFZOR-UHFFFAOYSA-N
Canonical SMILESCOc1ccc(-n2nc(C(C)C)cc2NC(=O)Nc2ccc(Oc3ccnc(Nc4cc(C)cc(C(=O)NCCN5CCOCC5)c4)n3)c3ccccc23)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.4
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P12931 SRC Homo sapiens Human PF07714 PF00017 PF00018 8.4 IC50 ChEMBL;BindingDB
Q16539 MAPK14 Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB