Molecule Details
InChIKeyWLQXBRYTQYYCMW-REWPJTCUSA-N
Compound Name(2S)-2-cyclopropyl-N-[(6S)-5,11-dioxospiro[3,6-dihydro-1H-pyrazolo[1,2-b][2,3]benzodiazepine-2,1'-cyclopropane]-6-yl]-N'-(5-fluoro-2-methylpyridin-3-yl)butanediamide
Canonical SMILESCc1ncc(F)cc1NC(=O)C[C@H](C(=O)N[C@@H]1C(=O)N2CC3(CC3)CN2C(=O)c2ccccc21)C1CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.74
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q8TCT8 SPPL2A Homo sapiens Human PF02225 PF04258 7.1 IC50 ChEMBL;BindingDB
Q8TCT7 SPPL2B Homo sapiens Human PF02225 PF04258 6.4 IC50 ChEMBL;BindingDB