Molecule Details
InChIKeyWLFMHNCEKPWCEA-UHFFFAOYSA-N
Compound Name1,6-Naphthyridine 37
Canonical SMILESCCN(CC)CCCCNc1cc2nc(NC(=O)NC(C)(C)C)c(-c3c(Cl)cccc3Cl)cc2cn1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.68
SourceBindingDB;ChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P12931 SRC Homo sapiens Human PF07714 PF00017 PF00018 7.8 IC50 BindingDB
P11362 FGFR1 Homo sapiens Human PF07679 PF00047 PF07714 7.6 pIC50 TTD_MultiTarget
P35968 KDR Homo sapiens Human PF07679 PF00047 PF13895 PF22971 PF07714 PF21339 PF17988 PF22854 7.6 IC50 ChEMBL;BindingDB