Molecule Details
InChIKeyWLBVZYXAXNRNOX-UHFFFAOYSA-N
Compound Name1-[3-Methoxy-6-[6-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]pyrazolo[4,3-c]pyridin-1-yl]pyridin-2-yl]-1,4-diazepan-6-ol
Canonical SMILESCOc1ccc(-n2ncc3cnc(-c4cnn(CC(F)(F)F)c4)cc32)nc1N1CCNCC(O)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.91
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 9.5 Ki ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 9.2 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.0 Ki ChEMBL;BindingDB