Molecule Details
InChIKeyWKWARMGSTJGPIX-UHFFFAOYSA-N
Compound Name6,11-Dihydropyridazino[4,3-c][1,5]benzodiazepin-5-one
Canonical SMILESO=C1Nc2ccccc2Nc2nnccc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.47
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49840 GSK3A Homo sapiens Human PF00069 6.7 Ki ChEMBL
O00444 PLK4 Homo sapiens Human PF00069 PF18190 PF18409 6.4 Ki ChEMBL
P48730 CSNK1D Homo sapiens Human PF00069 6.3 Ki ChEMBL