Molecule Details
InChIKeyWKUAOHBRCMZTIL-UHFFFAOYSA-N
Compound NameIndolocarbazole deriv. 12g
Canonical SMILESCOc1ccc2c3c4c(c5c(ccc6ccn(C)c65)c3n(CCCN3CCN(C)CC3)c2c1)C(=O)NC4=O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.71
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 7.8 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 7.8 pIC50 TTD_MultiTarget
P24385 CCND1 Homo sapiens Human PF02984 PF00134 7.4 IC50 ChEMBL