Molecule Details
InChIKeyWKPBGKVKFLTKJT-UHFFFAOYSA-N
Compound Name9-(4-methylpiperazin-1-yl)-7-[5-(trifluoromethyl)-1H-pyrazol-4-yl]-8,9,10,11-tetrahydro-3H-pyrazolo[4,5-a]phenanthridine
Canonical SMILESCN1CCN(C2CCc3c(c(-c4c[nH]nc4C(F)(F)F)nc4ccc5[nH]ncc5c34)C2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.67
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P36888 FLT3 Homo sapiens Human PF00047 PF07714 6.8 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 6.6 IC50 ChEMBL;BindingDB
P78396 CCNA1 Homo sapiens Human PF02984 PF00134 PF16500 6.6 IC50 ChEMBL