Molecule Details
InChIKeyWIWNZUYJVZDDEH-UHFFFAOYSA-N
Compound Name2-[({4-[(4-Tert-butylphenyl)methyl]piperazin-1-yl}sulfonyl)amino]-5-[(2-phenylethyl)sulfanyl]benzoic acid
Canonical SMILESCC(C)(C)c1ccc(CN2CCN(S(=O)(=O)Nc3ccc(SCCc4ccccc4)cc3C(=O)O)CC2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.57
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16548 BCL2A1 Homo sapiens Human PF00452 7.0 Ki ChEMBL;BindingDB
Q07820 MCL1 Homo sapiens Human PF00452 6.6 Ki ChEMBL;BindingDB
P55957 BID Homo sapiens Human PF06393 6.1 Ki ChEMBL