Molecule Details
InChIKeyWISKOZINSNUMIP-UHFFFAOYSA-N
Compound Name6-[[[4-Cyano-3-[2-(trifluoromethyl)phenyl]phenyl]-(3-methylimidazol-4-yl)methoxy]methyl]-2-(oxolan-2-ylmethylamino)pyridine-3-carbonitrile
Canonical SMILESCn1cncc1C(OCc1ccc(C#N)c(NCC2CCCO2)n1)c1ccc(C#N)c(-c2ccccc2C(F)(F)F)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.96
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 9.0 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 9.0 IC50 ChEMBL;BindingDB