Molecule Details
InChIKeyWIPBIZXEEPHOTH-UHFFFAOYSA-N
Compound NameN-methyl-5-[3-[4-(4-methylpiperazin-1-yl)pyrimidin-2-yl]-1H-indol-5-yl]-1,3,4-thiadiazol-2-amine
Canonical SMILESCNc1nnc(-c2ccc3[nH]cc(-c4nccc(N5CCN(C)CC5)n4)c3c2)s1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.94
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB