Molecule Details
InChIKeyWIIIHAKKVLVGJX-UHFFFAOYSA-N
Compound NamePyrazolo[1,5-b]pyridazine deriv. 27
Canonical SMILESc1cnn2ncc(-c3ccnc(Nc4ccc5c(c4)OCCO5)n3)c2c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.48
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49841 GSK3B Homo sapiens Human PF00069 9.0 IC50 ChEMBL;BindingDB
P11802 CDK4 Homo sapiens Human PF00069 8.2 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 8.2 pIC50 TTD_MultiTarget