Molecule Details
InChIKeyWHIABSZOSLXOTJ-UHFFFAOYSA-N
Compound Name1-[5-Ethyl-3-(pyrid-3-yl)phenylcarbamoyl]-5-methoxy6-trifluoromethylindoline
Canonical SMILESCCc1cc(NC(=O)N2CCc3cc(OC)c(C(F)(F)F)cc32)cc(-c2cccnc2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.97
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28335 HTR2C Homo sapiens Human PF00001 9.2 Ki ChEMBL;BindingDB
P41595 HTR2B Homo sapiens Human PF00001 8.0 Ki ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 6.7 Ki ChEMBL;BindingDB