Molecule Details
InChIKeyWHBHHAKSCKVYCJ-UHFFFAOYSA-N
Compound NameN-(2,3-Dimethylphenyl)-2-((3-(2-hydroxyphenyl)-1H-1,2,4-triazol-5-yl)thio)acetamide
Canonical SMILESCc1cccc(NC(=O)CSc2n[nH]c(-c3ccccc3O)n2)c1C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.17
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15118 PDK1 Homo sapiens Human PF10436 PF02518 6.3 IC50 ChEMBL;BindingDB
P07900 HSP90AA1 Homo sapiens Human PF13589 PF00183 6.1 IC50 ChEMBL
P08238 HSP90AB1 Homo sapiens Human PF13589 PF00183 6.1 IC50 ChEMBL;BindingDB