Molecule Details
InChIKeyWGYAMRMJVUNILQ-UHFFFAOYSA-N
Compound Name6-Chloro-4-phenyl-3-(5-phenyl-4,5-dihydro-1H-pyrazol-3-yl)quinolin-2(1H)-one
Canonical SMILESO=c1[nH]c2ccc(Cl)cc2c(-c2ccccc2)c1C1=NNC(c2ccccc2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.57
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q5VT25 CDC42BPA Homo sapiens Human PF00130 PF00780 PF08826 PF15796 PF25346 PF00069 PF00433 7.0 Ki ChEMBL
P28482 MAPK1 Homo sapiens Human PF00069 6.7 Ki ChEMBL
P17612 PRKACA Homo sapiens Human PF00069 6.0 Ki ChEMBL