Molecule Details
InChIKeyWGVPSTQRQHGEEP-UHFFFAOYSA-N
Compound NameN-{4-[2-(Dimethylamino)-1-(1H-imidazol-1-yl)propyl]phenyl}-1,3-benzothiazol-2-amine
Canonical SMILESCC(C(c1ccc(Nc2nc3ccccc3s2)cc1)n1ccnc1)N(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.93
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9NR63 CYP26B1 Homo sapiens Human PF00067 8.5 IC50 ChEMBL;BindingDB
O43174 CYP26A1 Homo sapiens Human PF00067 8.4 IC50 ChEMBL;BindingDB
P08684 CYP3A4 Homo sapiens Human PF00067 6.9 IC50 ChEMBL;BindingDB