Molecule Details
InChIKeyWGFMMFHWGQNJEB-UHFFFAOYSA-N
Compound Name5-fluoro-2-[4-methoxy-3-[2-(4-methylpiperidin-1-yl)ethoxy]phenyl]-7-(trifluoromethyl)-3H-isoindol-1-one
Canonical SMILESCOc1ccc(N2Cc3cc(F)cc(C(F)(F)F)c3C2=O)cc1OCCN1CCC(C)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.53
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28335 HTR2C Homo sapiens Human PF00001 9.4 Ki ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 6.6 Ki ChEMBL;BindingDB
P41595 HTR2B Homo sapiens Human PF00001 6.6 Ki ChEMBL;BindingDB