Molecule Details
InChIKeyWFXRLISEEGXGJM-UHFFFAOYSA-N
Compound NameUS11377423, Cmpd 2A
Canonical SMILESNc1cc(F)ccc1NC(=O)c1ccc(CNc2nccc(-c3cccnc3)n2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.81
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13547 HDAC1 Homo sapiens Human PF00850 7.9 IC50 ChEMBL;BindingDB
O15379 HDAC3 Homo sapiens Human PF00850 7.8 IC50 BindingDB
Q92769 HDAC2 Homo sapiens Human PF00850 7.7 IC50 BindingDB