Molecule Details
InChIKeyWFRCVVPACDUWGD-BUDLEJPASA-N
Canonical SMILESO=C(O)CN(CCc1ccccc1)C(=O)C(Cc1c[nH]c2ccccc12)NC(=O)OC1[C@H]2C[C@@H]3C[C@@H](C[C@H]1C3)C2
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.65
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P32238 CCKAR Homo sapiens Human PF00001 PF09193 6.7 pIC50 TTD_MultiTarget
P32239 CCKBR Homo sapiens Human PF00001 6.7 Ki ChEMBL