Molecule Details
InChIKeyWETYFBSRFBUFCI-KSMSDSDGSA-N
Compound Name(3R,4S)-N-[(2R)-4-[6-(4-chlorophenyl)sulfanyl-2-(4-methoxyphenyl)-3-oxopyridazin-4-yl]butan-2-yl]-4-(4-fluorophenyl)piperidine-3-carboxamide
Canonical SMILESCOc1ccc(-n2nc(Sc3ccc(Cl)cc3)cc(CC[C@@H](C)NC(=O)[C@H]3CNCC[C@@H]3c3ccc(F)cc3)c2=O)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.69
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P32245 MC4R Homo sapiens Human PF00001 8.0 IC50 ChEMBL;BindingDB
P33032 MC5R Homo sapiens Human PF00001 6.1 IC50 ChEMBL;BindingDB
P41968 MC3R Homo sapiens Human PF00001 6.0 IC50 ChEMBL;BindingDB