Molecule Details
InChIKeyWEMGUFBETKXSRV-UHFFFAOYSA-N
Compound NameN'-hydroxy-2-(3-imidazo[1,2-a]pyridin-2-ylphenyl)-3H-benzimidazole-5-carboximidamide
Canonical SMILESN=C(NO)c1ccc2nc(-c3cccc(-c4cn5ccccc5n4)c3)[nH]c2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.43
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08684 CYP3A4 Homo sapiens Human PF00067 6.6 IC50 ChEMBL;BindingDB
Q92769 HDAC2 Homo sapiens Human PF00850 6.4 IC50 ChEMBL;BindingDB
Q13547 HDAC1 Homo sapiens Human PF00850 6.3 IC50 ChEMBL;BindingDB