Molecule Details
InChIKeyWDUJNEUBVHIQQH-CQSZACIVSA-N
Compound Name(6aR)-4-(cyclobutylmethyl)-6,6a,7,8,9,10-hexahydro-5H-pyrazino[1,2-a][1,8]naphthyridine
Canonical SMILESc1cc(CC2CCC2)c2c(n1)N1CCNC[C@H]1CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.69
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28223 HTR2A Homo sapiens Human PF00001 7.9 Ki ChEMBL;BindingDB
P28335 HTR2C Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB
P41595 HTR2B Homo sapiens Human PF00001 7.4 Ki ChEMBL;BindingDB