Molecule Details
InChIKeyWDTMXLCGAKGDKL-UHFFFAOYSA-N
Compound Name9-(3-Hydroxy-3-methyl-but-1-ynyl)-4,5-dihydro-[1]benzoxepino[5,4-d]thiazole-2-carboxamide
Canonical SMILESCC(C)(O)C#Cc1ccc2c(c1)-c1nc(C(N)=O)sc1CCO2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.95
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q99558 MAP3K14 Homo sapiens Human PF00069 7.5 Ki ChEMBL;BindingDB
O00329 PIK3CD Homo sapiens Human PF00454 PF00792 PF02192 PF00794 PF00613 6.7 Ki ChEMBL
P27986 PIK3R1 Homo sapiens Human PF16454 PF00620 PF00017 6.7 Ki ChEMBL;BindingDB