Molecule Details
InChIKeyWDNVNCPECUHEGM-DODPDUHYSA-N
Compound NameUS10807971, Example 17
Canonical SMILESN[C@H]1C[C@@H](N2CC=C(c3ncc(N4CC[C@](O)(C(=O)NCc5cc(F)cc(Cl)c5)C4=O)cn3)CC2)CO[C@@H]1c1cc(F)ccc1F
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.1
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P27487 DPP4 Homo sapiens Human PF00930 PF00326 7.8 IC50 ChEMBL;BindingDB
P50579 METAP2 Homo sapiens Human PF00557 6.4 IC50 ChEMBL;BindingDB