Molecule Details
InChIKeyWDIPTEIUSFFSDV-WEMQTCASSA-N
Compound Name(2E,4E,6E)-3-Methyl-6-fluoro-7-[2-(2,2-difluoroethoxy)-3,5-di-tert-butylphenyl]-2,4,6-octatrienoic acid
Canonical SMILESCC(/C=C/C(F)=C(/C)c1cc(C(C)(C)C)cc(C(C)(C)C)c1OCC(F)F)=C\C(=O)O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.97
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P19793 RXRA Homo sapiens Human PF00104 PF11825 PF00105 8.1 Ki ChEMBL;BindingDB
P28702 RXRB Homo sapiens Human PF00104 PF00105 7.9 Ki ChEMBL;BindingDB
P48443 RXRG Homo sapiens Human PF00104 PF11825 PF00105 7.9 Ki ChEMBL;BindingDB