Molecule Details
InChIKeyWDCPMDKQCCZVEW-VMPITWQZSA-N
Compound Name7-Methoxy-3-[4-((E)-3-phenyl-allyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-chromeno[4,3-c]isoxazole
Canonical SMILESCOc1ccc2c(c1)OCC1C2=NOC1CN1CCN(C/C=C/c2ccccc2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.61
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08913 ADRA2A Homo sapiens Human PF00001 9.3 Ki ChEMBL;BindingDB
P18825 ADRA2C Homo sapiens Human PF00001 8.7 Ki ChEMBL;BindingDB
P18089 ADRA2B Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB