Molecule Details
InChIKeyWCTNEALHPXRJMI-UHFFFAOYSA-N
Compound Name3-((4-((4-(3-(3-isopropyl-1-(p-tolyl)-1H-pyrazol-5-yl)ureido)naphthalen-1-yl)oxy)pyrimidin-2-yl)amino)-4-methoxy-N-(2-morpholinoethyl)benzamide
Canonical SMILESCOc1ccc(C(=O)NCCN2CCOCC2)cc1Nc1nccc(Oc2ccc(NC(=O)Nc3cc(C(C)C)nn3-c3ccc(C)cc3)c3ccccc23)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.17
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P12931 SRC Homo sapiens Human PF07714 PF00017 PF00018 9.0 IC50 ChEMBL;BindingDB
Q16539 MAPK14 Homo sapiens Human PF00069 8.5 IC50 ChEMBL;BindingDB
P43405 SYK Homo sapiens Human PF07714 PF00017 7.0 IC50 ChEMBL;BindingDB