Molecule Details
InChIKeyWCOSWMKQOOTINK-UHFFFAOYSA-N
Compound Name2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-isobutyl-1H-indol-4-yloxy)acetic acid
Canonical SMILESCC(C)Cc1c(C(=O)C(N)=O)c2c(OCC(=O)O)cccc2n1Cc1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.62
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O15496 PLA2G10 Homo sapiens Human PF00068 7.3 IC50 ChEMBL;BindingDB
Q9UNK4 PLA2G2D Homo sapiens Human PF00068 6.3 IC50 ChEMBL;BindingDB
Q9BZM2 PLA2G2F Homo sapiens Human PF00068 6.3 IC50 ChEMBL;BindingDB