Molecule Details
InChIKeyWCJKXYDSZKCXFG-GEPWALDNSA-N
Canonical SMILESCOc1cc(OC)cc([C@@H](C(=O)N2CCCC[C@H]2C(=O)O[C@H](CCc2ccc(OC)c(OC)c2)c2cccc(OCC(=O)O)c2)C2CCCCC2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.59
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13451 FKBP5 Homo sapiens Human PF00254 PF00515 PF13181 7.0 Ki ChEMBL;BindingDB
P62942 FKBP1A Homo sapiens Human PF00254 6.2 Ki ChEMBL;BindingDB