Molecule Details
InChIKeyWCHWFNCOZFCZSO-UHFFFAOYSA-N
Compound Name1-[5-(4-Fluoro-phenyl)-pyridin-3-ylmethyl]-4-pyridin-2-yl-piperazine
Canonical SMILESFc1ccc(-c2cncc(CN3CCN(c4ccccn4)CC3)c2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.3
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P21917 DRD4 Homo sapiens Human PF00001 8.2 IC50 ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 7.2 IC50 ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 6.5 IC50 ChEMBL;BindingDB