Molecule Details
InChIKeyWCEHIDWONYOKOJ-UHFFFAOYSA-N
Compound NamePROTAC CDK9 Degrader-1
Canonical SMILESO=C1CCC(N2C(=O)c3cccc(OCCCCCOc4ccc(CC(=O)Nc5cc(C6CCC6)[nH]n5)cc4)c3C2=O)C(=O)N1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.21
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96SW2 CRBN Homo sapiens Human PF02190 PF03226 7.4 IC50 ChEMBL
P24941 CDK2 Homo sapiens Human PF00069 7.1 IC50 ChEMBL
Q00535 CDK5 Homo sapiens Human PF00069 7.1 IC50 ChEMBL