Molecule Details
InChIKeyWBPFBRSQEAARNO-UHFFFAOYSA-N
Compound Name4-(1-isopropyl-2-methyl-1H-imidazol-5-yl)-N-(4-(2-methoxyethylsulfonyl)phenyl)pyrimidin-2-amine
Canonical SMILESCOCC[S@SP3](=O)(=O)c1ccc(Nc2nccc(-c3cnc(C)n3C(C)C)n2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.85
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 7.8 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 7.8 pIC50 TTD_MultiTarget