Molecule Details
InChIKeyWBFASLOAEQLKGO-UHFFFAOYSA-N
Compound Name[2,3-Dihydro-8-(4-methyl-1-piperazinyl)-1H-pyrrolo[3,2-g]isoquinolin-1-yl]-5-quinolinylmethanone
Canonical SMILESCN1CCN(c2nccc3cc4c(cc23)N(C(=O)c2cccc3ncccc23)CC4)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.63
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28222 HTR1B Homo sapiens Human PF00001 9.1 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 8.4 Ki ChEMBL;BindingDB
P28221 HTR1D Homo sapiens Human PF00001 8.4 Ki ChEMBL;BindingDB