Molecule Details
InChIKeyWBBBVZGQADABSU-VPUGGFGBSA-N
Compound NameAc-Arg-Tyr-Tyr-Arg-D-aIle-Lys-NH2
Canonical SMILESCC[C@H](C)[C@@H](NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CCCNC(=N)N)NC(C)=O)C(=O)N[C@@H](CCCCN)C(N)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.3
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P41146 OPRL1 Homo sapiens Human PF00001 9.3 Ki ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB
P41145 OPRK1 Homo sapiens Human PF00001 6.1 Ki ChEMBL;BindingDB