Molecule Details
InChIKeyWAOZMJFYNREQLU-MJWYEJTISA-N
Canonical SMILESCOc1cc(N2CCN(CCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)(C)C)CC2)ccc1NC(=O)c1cccc(-c2cc[nH]n2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.76
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P51617 IRAK1 Homo sapiens Human PF00531 PF00069 7.1 IC50 ChEMBL;BindingDB
Q9NWZ3 IRAK4 Homo sapiens Human PF07714 6.4 IC50 ChEMBL;BindingDB