Molecule Details
InChIKeyWAKJOUVIVRSNKI-UHFFFAOYSA-N
Compound Name1,3-dihydroisoindol-2-yl-[6-hydroxy-3-[(3-methylphenyl)methyl]-2H-indazol-5-yl]methanone
Canonical SMILESCc1cccc(Cc2n[nH]c3cc(O)c(C(=O)N4Cc5ccccc5C4)cc23)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.25
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49336 CDK8 Homo sapiens Human PF00069 7.8 IC50 ChEMBL
P07900 HSP90AA1 Homo sapiens Human PF13589 PF00183 7.0 IC50 ChEMBL
P08238 HSP90AB1 Homo sapiens Human PF13589 PF00183 7.0 IC50 ChEMBL