Molecule Details
InChIKeyVZXFJJIXYUECLL-UHFFFAOYSA-N
Compound Name2-(4-Fluorophenyl)-3-(2-methylsulfanylpyrimidin-4-yl)imidazo[1,2-a]pyrazin-8-amine
Canonical SMILESCSc1nccc(-c2c(-c3ccc(F)cc3)nc3c(N)nccn23)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.25
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49674 CSNK1E Homo sapiens Human PF00069 6.7 IC50 ChEMBL;BindingDB
Q00535 CDK5 Homo sapiens Human PF00069 6.0 IC50 ChEMBL
Q15078 CDK5R1 Homo sapiens Human PF03261 6.0 IC50 ChEMBL;BindingDB