Molecule Details
InChIKeyVZRKGDOTBQOIIT-LQJZCPKCSA-N
Compound Name{1-[2-Oxo-1-phenethyl-3-(3-phenyl-propylsulfanyl)-propylcarbamoyl]-2-phenyl-ethyl}-carbamic acid pyridin-3-ylmethyl ester
Canonical SMILESO=C(N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCc1ccccc1)C(=O)CSCCCc1ccccc1)OCc1cccnc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.58
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P07711 CTSL Homo sapiens Human PF08246 PF00112 7.5 Ki ChEMBL;BindingDB
P07858 CTSB Homo sapiens Human PF00112 PF08127 6.2 Ki ChEMBL;BindingDB
P25779 Trypanosoma cruzi Pathogen PF12131 PF08246 PF00112 9.1 Ki ChEMBL;BindingDB