Molecule Details
InChIKeyVZBQJKIOAOUYJL-UHFFFAOYSA-N
Compound Name(1-Methyl-1h-Imidazol-2-Yl)-(3-Methyl-4-(3-((Pyridin-3-Ylmethyl)-Amino)-Propoxy)-Benzofuran-2-Yl)-Methanone
Canonical SMILESCc1c(C(=O)c2nccn2C)oc2cccc(OCCCNCc3cccnc3)c12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.89
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB03062
Drug Name(1-Methyl-1h-Imidazol-2-Yl)-(3-Methyl-4-{3-[(Pyridin-3-Ylmethyl)-Amino]-Propoxy}-Benzofuran-2-Yl)-Methanone
CAS Numbernan
Groups experimental
ATC Codes nan
Descriptionnan

Categories: Dietary Supplements Supplements
Cross-references: BindingDB: 50121720 CHEMBL355497 ChemSpider: 393760 PDB: R64 PubChem:446386 PubChem:46505140 ZINC: ZINC000003581083
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O60551 NMT2 Homo sapiens Human PF01233 PF02799 8.9 IC50 ChEMBL
P30419 NMT1 Homo sapiens Human PF01233 PF02799 8.9 IC50 ChEMBL;BindingDB
DrugBank Target Actions (2)
Target Gene Target Name Action Type
P30418 NMT1 Glycylpeptide N-tetradecanoyltransferase binder targets
P30419 NMT1 Glycylpeptide N-tetradecanoyltransferase 1 binder targets