Molecule Details
InChIKeyVYVLVTDHSCQXGE-UHFFFAOYSA-N
Compound NameN-methyl-6-[6-(6-methylpyrazin-2-yl)pyrazolo[4,3-c]pyridin-1-yl]pyridin-2-amine
Canonical SMILESCNc1cccc(-n2ncc3cnc(-c4cncc(C)n4)cc32)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.15
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 9.6 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 9.4 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.5 Ki ChEMBL;BindingDB