Molecule Details
InChIKeyVYTQMUCONGRNBX-UHFFFAOYSA-N
Compound Namedimethyl-{2-[(4-{4-[3-(pyridin-2-yl)-1H-pyrazol-4-yl]-2-pyridinyl}phenyl)oxy]ethyl}amine
Canonical SMILESCN(C)CCOc1ccc(-c2cc(-c3c[nH]nc3-c3ccccn3)ccn2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.63
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P36897 TGFBR1 Homo sapiens Human PF01064 PF00069 PF08515 7.8 IC50 ChEMBL;BindingDB
P01137 TGFB1 Homo sapiens Human PF00019 PF00688 7.7 IC50 BindingDB
P36896 ACVR1B Homo sapiens Human PF01064 PF00069 PF08515 7.3 IC50 ChEMBL