Molecule Details
InChIKeyVYQHPOVDIRILEA-UHFFFAOYSA-N
Compound NameMethyl 4-methyl-2-(2-(2-oxo-3,4-dihydroquinolin-1(2H)-yl)acetamido)thiophene-3-carboxylate
Canonical SMILESCOC(=O)c1c(C)csc1NC(=O)CN1C(=O)CCc2ccccc21
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.72
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 6.9 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 6.2 IC50 ChEMBL;BindingDB